Oxabolone cipionate |
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| Trade names | Steranabol Depo, Steranabol Ritardo |
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| Other names | Oxabolone cypionate; FI-5852; 4-Hydroxy-19-nortestosterone 17β-cypionate; Estr-4-en-4,17β-diol-3-one 17β-cypionate |
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Routes of administration | Intramuscular injection[1] |
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| Drug class | Androgen; Anabolic steroid; Androgen ester |
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| ATC code | |
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[(8R,9S,10R,13S,14S,17S)-4-hydroxy-13-methyl-3-oxo-2,6,7,8,9,10,11,12,14,15,16,17-dodecahydro-1H-cyclopenta[a]phenanthren-17-yl]-3-cyclopentylpropanoate
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| ECHA InfoCard | 100.013.647 |
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| Formula | C26H38O4 |
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| Molar mass | 414.586 g·mol−1 |
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| 3D model (JSmol) | |
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C[C@]12CC[C@H]3[C@H]([C@@H]1CC[C@@H]2OC(=O)CCC4CCCC4)CCC5=C(C(=O)CC[C@H]35)O
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InChI=1S/C26H38O4/c1-26-15-14-18-17-9-11-22(27)25(29)20(17)8-7-19(18)21(26)10-12-23(26)30-24(28)13-6-16-4-2-3-5-16/h16-19,21,23,29H,2-15H2,1H3/t17-,18-,19-,21+,23+,26+/m1/s1 NKey:KHKDIUPVDIEHAH-KXLSUQFWSA-N N
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N Y (what is this?) (verify) |
Oxabolone cipionate (INNTooltip International Nonproprietary Name, JANTooltip Japanese Accepted Name) (brand names Steranabol Depo, Steranabol Ritardo; former developmental code name FI-5852), or oxabolone cypionate, also known as 4-hydroxy-19-nortestosterone 17β-cypionate or estr-4-en-4,17β-diol-3-one 17β-cypionate, is synthetic and injected anabolic–androgenic steroid (AAS) and derivative of nandrolone (19-nortestosterone) which has been marketed in Europe.[1][2][3] It is the C17β cypionate ester and a prodrug of oxabolone (4-hydroxy-19-nortestosterone).[2][3]
See also
- 4-Hydroxytestosterone
- Clostebol (4-chlorotestosterone)
- Formestane (4-hydroxyandrostenedione)
- Norclostebol (4-chloro-19-nortestosterone)
References
Androgens and antiandrogens |
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Androgens (incl. AASTooltip anabolic–androgenic steroid) | | ARTooltip Androgen receptor agonists |
- Dihydrotestosterone derivatives: Androstanolone (stanolone, dihydrotestosterone, DHT)
- Androstanolone esters
- Bolazine capronate
- Drostanolone propionate (dromostanolone propionate)
- Epitiostanol
- Mepitiostane
- Mesterolone
- Metenolone acetate (methenolone acetate)
- Metenolone enanthate (methenolone enanthate)
- Stenbolone acetate
- 19-Nortestosterone derivatives: Bolandiol dipropionate
- Nandrolone esters (e.g., nandrolone decanoate, nandrolone phenylpropionate)
- Norclostebol
- Norclostebol acetate
- Oxabolone cipionate (oxabolone cypionate)
- Trenbolone acetate
- Trenbolone hexahydrobenzylcarbonate (trenbolone cyclohexylmethylcarbonate)
- 17α-Alkylated 19-nortestosterone derivatives: Ethylestrenol
- Mibolerone
- Norethandrolone
- Normethandrone (methylestrenolone, normethisterone)
- Propetandrol (propethandrol)
- 17α-Vinyltestosterone derivatives: Norvinisterone (vinylnortestosterone)
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| Progonadotropins |
- Antiestrogens (e.g., tamoxifen, clomifene)
- GnRH agonists (e.g., GnRH (gonadorelin), leuprorelin)
- Gonadotropins (e.g., LHTooltip luteinizing hormone, hCGTooltip human chorionic gonadotropin)
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| Antiandrogens | | ARTooltip Androgen receptor antagonists |
- Steroidal: Abiraterone acetate +niraparib
- Canrenone
- Chlormadinone acetate
- Cyproterone acetate
- Delmadinone acetate
- Dienogest
- Drospirenone
- Medrogestone
- Megestrol acetate
- Nomegestrol acetate
- Osaterone acetate
- Oxendolone
- Potassium canrenoate
- Spironolactone
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Steroidogenesis inhibitors | |
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| Antigonadotropins |
- D2 receptor antagonists (prolactin releasers) (e.g., domperidone, metoclopramide, risperidone, haloperidol, chlorpromazine, sulpiride)
- Estrogens (e.g., bifluranol, diethylstilbestrol, estradiol, estradiol esters, ethinylestradiol, ethinylestradiol sulfonate, paroxypropione)
- GnRH agonists (e.g., leuprorelin)
- GnRH antagonists (e.g., cetrorelix)
- Progestogens (incl., chlormadinone acetate, cyproterone acetate, hydroxyprogesterone caproate, gestonorone caproate, medroxyprogesterone acetate, megestrol acetate)
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| Others | |
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- #WHO-EM
- ‡Withdrawn from market
- Clinical trials:
- †Phase III
- §Never to phase III
- See also
- Androgen receptor modulators
- Estrogens and antiestrogens
- Progestogens and antiprogestogens
- List of androgens/anabolic steroids
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Androgen receptor modulators |
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| ARTooltip Androgen receptor | | Agonists | |
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| SARMsTooltip Selective androgen receptor modulator |
- Nonsteroidal: 198RL26
- ACP-105
- AC-262,536
- Acetothiolutamide
- Acetoxolutamide
- Andarine (acetamidoxolutamide, androxolutamide, GTx-007, S-4)
- BMS-564,929
- DTIB
- Enobosarm (ostarine, MK-2866, GTx-024, S-22)
- FTBU-1
- GLPG-0492
- GSK2881078
- GSK-4336A
- GSK-8698
- LG121071 (LGD-121071)
- LGD-2226
- LGD-2941 (LGD-122941)
- LGD-3303
- LGD-4033
- LY305
- JNJ-26146900
- JNJ-28330835
- JNJ-37654032
- OPK-88004 (LY-2452473, TT-701)
- ORM-11984
- PF-06260414
- R-1
- RU-59063
- S-1
- S-23
- S-40503
- S-101479
- Vosilasarm
- Steroidal: EM-9017
- MK-0773
- S42
- TFM-4AS-1
- YK-11
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| Antagonists |
- Steroidal: 7α-Thioprogesterone
- 7α-Thiospironolactone
- 7α-Thiomethylspironolactone
- 11α-Hydroxyprogesterone
- 15β-Hydroxycyproterone acetate
- Abiraterone
- Abiraterone acetate
- Allyltestosterone
- Benorterone
- BOMT
- Canrenoic acid
- Canrenone
- Chlormadinone acetate
- Clascoterone
- Clometerone
- Cyproheptadine
- Cyproterone
- Cyproterone acetate
- Delanterone
- Delmadinone acetate
- Dicirenone
- Dienogest
- Drospirenone
- DU-41165
- Edogestrone
- EM-4350
- EM-5854
- EM-5855
- EM-6537
- Epitestosterone
- Galeterone
- Guggulsterone
- Ludaterone
- Medrogestone
- Megestrol acetate
- Mespirenone
- Metogest
- Mexrenone
- Mifepristone
- Nomegestrol acetate
- Nordinone
- Osaterone
- Osaterone acetate
- Oxendolone
- Potassium canrenoate
- Promegestone
- Prorenone
- Rosterolone
- RU-15328
- SC-5233 (spirolactone)
- Spironolactone
- Spirorenone
- Spiroxasone
- Topterone
- Trimegestone
- Trimethyltrienolone (R-2956)
- Zanoterone
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| GPRC6A | |
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- See also
- Receptor/signaling modulators
- Androgens and antiandrogens
- Estrogen receptor modulators
- Progesterone receptor modulators
- List of androgens and anabolic steroids
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